Inventors:
Xianchang Gong - La Jolla CA, US
Kathy Barrett - La Jolla CA, US
Jianguo Cao - San Diego CA, US
Colleen Gritzen - Vista CA, US
Glenn Noronha - Seattle WA, US
John D. Hood - San Diego CA, US
Chi Ching Mak - San Diego CA, US
Andrew McPherson - San Diego CA, US
Ved Prakash Pathak - San Diego CA, US
Joel Renick - San Diego CA, US
Richard M. Soll - San Diego CA, US
Ute Splittgerber - South San Francisco CA, US
Wolfgang Wrasidlo - La Jolla CA, US
Binqi Zeng - San Diego CA, US
Ningning Zhao - San Diego CA, US
Elena Dneprovskaia - San Diego CA, US
Assignee:
TargeGen, Inc. - Bridgewater NJ
International Classification:
A61K 31/53
A61P 35/00
C07D 401/12
C07D 401/14
C07D 403/04
C07D 403/12
C07D 403/14
C07D 413/12
C07D 413/14
C07D 417/12
C07D 417/14
Abstract:
The invention provides benzotriazine compounds having formula (I). The benzotriazine compounds of the invention are capable of inhibiting kinases, such members of the Src kinase family, and various other specific receptor and non-receptor kinases.